Structure
CV-6209, Inhibitor
CV-6209
Purity
>98% (HPLC)
Synonyms
CV-6209; CV 6209; CV6209; inhibitor
Purity/Purification
>98% (HPLC)
Target
Platelet-activating Factor Receptor
Receptor
Platelet-activating Factor Receptor
Chemical Name
2-[N-acetyl-N-(2-methoxy-3-octadecylcarbamoyloxypropoxycarbonyl) aminomethyl]-1-ethylpyridinium chloride
SMILES
O=C(OCC(OC)COC(N(C(C)=O)CC1=CC=CC=[N+]1CC)=O)NCCCCCCCCCCCCCCCCCC
Molecular Formula
C34H60N3O6Cl
CAS Number
100488-87-7
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Stability: >=2 years
Shipping: Ice Pack
Structure
Structure
Related Product Information for CV-6209, inhibitor
A highly potent, selective platelet activating factor (PAF) inhibitor with IC50 of 75 and 170nM for aggregation inhibition of rabbit and human platelets induced by PAF; shows little to no effects on the aggregation induced by arachidonic acid, ADP and collagen; inhibited PAF-induced hypotension in rats (ED50=0.009mg/kg i.v.) with no effect on the hypotension induced by arachidonic acid, histamine, bradykinin and isoproterenol. Ulcer Discontinued
Product Categories/Family for CV-6209, inhibitor
References
1. Terashita Z, et al. J Pharmacol Exp Ther. 1987 Jul; 242 (1):263-8.
2. Terashita Z, et al. J Cardiovasc Pharmacol. 1988; 12 (5):505-11.
3. Stahl GL, et al. J Pharmacol Exp Ther. 1988 Mar; 244 (3):898-904.
4. Takatani M, et al. J Med Chem. 1989 Jan; 32 (1):56-64.
2. Terashita Z, et al. J Cardiovasc Pharmacol. 1988; 12 (5):505-11.
3. Stahl GL, et al. J Pharmacol Exp Ther. 1988 Mar; 244 (3):898-904.
4. Takatani M, et al. J Med Chem. 1989 Jan; 32 (1):56-64.
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Product Notes
The CV-6209 (Catalog #AAA3600036) is an Inhibitor and is intended for research purposes only. The product is available for immediate purchase. It is sometimes possible for the material contained within the vial of "CV-6209, Inhibitor" to become dispersed throughout the inside of the vial, particularly around the seal of said vial, during shipment and storage. We always suggest centrifuging these vials to consolidate all of the liquid away from the lid and to the bottom of the vial prior to opening. Please be advised that certain products may require dry ice for shipping and that, if this is the case, an additional dry ice fee may also be required.Precautions
All products in the AAA Biotech catalog are strictly for research-use only, and are absolutely not suitable for use in any sort of medical, therapeutic, prophylactic, in-vivo, or diagnostic capacity. By purchasing a product from AAA Biotech, you are explicitly certifying that said products will be properly tested and used in line with industry standard. AAA Biotech and its authorized distribution partners reserve the right to refuse to fulfill any order if we have any indication that a purchaser may be intending to use a product outside of our accepted criteria.Disclaimer
Though we do strive to guarantee the information represented in this datasheet, AAA Biotech cannot be held responsible for any oversights or imprecisions. AAA Biotech reserves the right to adjust any aspect of this datasheet at any time and without notice. It is the responsibility of the customer to inform AAA Biotech of any product performance issues observed or experienced within 30 days of receipt of said product. To see additional details on this or any of our other policies, please see our Terms & Conditions page.Item has been added to Shopping Cart
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