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25 results for "TrkA inhibitor" - showing 1-25
Structure
Danusertib, Inhibitor (Cat# AAA575889)
Full Name
Danusertib
Purity
98.4%
Pricing
$215/2 mg | $245/5 mg | $325/10 mg | $485/25 mg | $700/50 mg | $250/1 mL (in DMSO) | $2,875/5x50 mg
Lestaurtinib (KT5555), Inhibitor (Cat# AAA515053)
Full Name
Lestaurtinib (KT5555)
Pricing
$185/5 mg | $290/25 mg | $1,080/5x25 mg
Structure
GNF-5837, Inhibitor (Cat# AAA578670)
Full Name
GNF-5837
Purity
99.3%
Pricing
$180/2 mg | $195/5 mg | $225/10 mg | $265/25 mg | $325/50 mg | $440/100 mg | $540/200 mg | $200/1 mL (in DMSO) | $2,160/5x200 mg
Testing Data
(PHA-793887 is a novel pan-cdk inhibitor, including cdk1, cdk2, cdk4, cdk5, cdk7, and cdk9 with IC50 in the 5 to 140 nM range. [1]It is inactive against other 34 kinases representative of all kinase families, in particular c-abl, c-kit, lck, and TRKA with IC50>10 mM. It shows anti-proliferative activity against several solid tumor cell lines, with IC50, 1 mM. In these cells, it is able to inhibit Rb phosphorylation and expression of S-phase cyclins, such as cyclin A. [1,2])
Chemical Structure
(Chemical structure of Lestaurtinib (SIH-460), a FLT3/ TrkA kinase inhibitor. CAS #: 111358-88-4. Molecular Formula: C26H21N3O4. Molecular Weight: 439.5 g/mol.)
Lestaurtinib, Small Molecule (Cat# AAA808160)
Full Name
Lestaurtinib
Purity
>=98% (HPLC)
Pricing
$280/1 mg | $630/5 mg | $1,015/5x1 mg | $2,600/5x5 mg
Structure
BMS-754807, Inhibitor (Cat# AAA3600014)
Full Name
BMS-754807
Purity
>98% (HPLC)
Pricing
$190/2 mg | $205/5 mg | $240/10 mg | $345/25 mg | $500/50 mg | $750/100 mg | $3,100/5x100 mg
Structure
DS-6051b, Inhibitor (Cat# AAA5756839)
Full Name
DS-6051b
Purity
98.00%
Pricing
$275/2 mg | $330/5 mg | $425/10 mg | $665/25 mg | $925/50 mg | $1,325/100 mg | $1,930/200 mg | $8,420/5x200 mg
Structure
AZ-23, Inhibitor (Cat# AAA5754554)
Full Name
AZ-23
Purity
98.00%
Pricing
$240/2 mg | $275/5 mg | $340/10 mg | $570/25 mg | $880/50 mg | $1,415/100 mg | $285/1mL*10mM (in DMSO) | $6,085/5x100 mg
Structure
GNF-5837, Inhibitor (Cat# AAA3607758)
Full Name
GNF-5837
Purity
>98% (HPLC)
Pricing
$190/2 mg | $210/5 mg | $235/10 mg | $295/25 mg | $375/50 mg | $555/100 mg | $715/200 mg | $2,945/5x200 mg
Structure
URMC-099, Inhibitor (Cat# AAA3600902)
Full Name
URMC-099
Purity
>98% (HPLC)
Pricing
$200/5 mg | $215/10 mg | $265/25 mg | $335/50 mg | $480/100 mg | $1,870/5x100 mg
Structure
PF-03814735, Inhibitor (Cat# AAA3607673)
Full Name
PF-03814735
Purity
>98% (HPLC)
Pricing
$690/50 mg | $2,825/5x50 mg
Structure
GW 441756, Inhibitor (Cat# AAA3607521)
Full Name
GW 441756
Purity
>98% (HPLC)
Pricing
$190/5 mg | $215/10 mg | $295/25 mg | $395/50 mg | $615/100 mg | $2,480/5x100 mg
Structure
Tavilermide, Inhibitor (Cat# AAA5755591)
Full Name
Tavilermide
Purity
98.00%
Pricing
$275/1 mg | $510/5 mg | $765/10 mg | $2,035/50 mg | $2,910/100 mg | $12,800/5x100 mg
Structure
RIPK1-IN-7, Inhibitor (Cat# AAA5753826)
Full Name
RIPK1-IN-7
Purity
98.00%
Pricing
$515/5 mg | $765/10 mg | $2,035/50 mg | $2,905/100 mg | $550/1 mL (in DMSO) | $12,805/5x100 mg
Chemical Structure
AZ 23, Inhibitor (Cat# AAA387367)
Full Name
AZ 23
Purity
>98%
Pricing
$225/5 mg | $320/10 mg | $630/25 mg | $1,055/50 mg | $4,680/5x50 mg
Ensartinib dihydrochloride, Inhibitor (Cat# AAA5756843)
Full Name
Ensartinib dihydrochloride
Purity
98.00%
Pricing
$245/2 mg | $330/5 mg | $1,210/5x5 mg
Structure
Lestaurtinib, Inhibitor (Cat# AAA5755089)
Full Name
Lestaurtinib
Purity
98.00%
Pricing
$715/5 mg | $700/1mL*10mM (in DMSO) | $2,925/5x5 mg
Structure
Danusertib, Inhibitor (Cat# AAA3606070)
Full Name
Danusertib
Purity
>98% (HPLC)
Pricing
$210/2 mg | $240/5 mg | $310/10 mg | $445/25 mg | $640/50 mg | $2,600/5x50 mg
Chemical Structure
GW 441756, Inhibitor (Cat# AAA3841506)
Full Name
GW 441756
Purity
>98%
Pricing
$160/10 mg | $375/50 mg | $1,625/5x50 mg
CE-245677, Inhibitor (Cat# AAA3843832)
Full Name
CE-245677
Purity
>98%
Pricing
$420/1 mg | $1,155/5 mg | $1,900/10 mg | $8,485/5x10 mg
Belizatinib, Inhibitor (Cat# AAA3845356)
Full Name
Belizatinib
Purity
>98%
Pricing
$135/2 mg | $190/5 mg | $295/10 mg | $760/50 mg | $3,385/5x50 mg
Testing Data
Lestaurtinib, Inhibitor (Cat# AAA516368)
Full Name
Lestaurtinib
Purity
>98% (TLC); NMR (Conforms)
Pricing
$255/1 mg | $645/5 mg | $2,685/5x5 mg
Structure
CH7057288, Inhibitor (Cat# AAA5751992)
Full Name
CH7057288
Purity
98.00%
Pricing
$245/2 mg | $360/5 mg | $570/10 mg | $985/25 mg | $1,485/50 mg | $2,270/100 mg | $9,940/5x100 mg
Structure
Selitrectinib, Inhibitor (Cat# AAA5758331)
Full Name
Selitrectinib
Purity
98.00%
Pricing
$195/1 mg | $230/5 mg | $265/10 mg | $360/25 mg | $480/50 mg | $800/100 mg | $230/1 mL (in DMSO) | $3,340/5x100 mg
Structure
PHA-848125, Inhibitor (Cat# AAA3606002)
Full Name
PHA-848125
Purity
>98% (HPLC)
Pricing
$435/10 mg | $930/50 mg | $3,900/5x50 mg
