Structure
GSK5182 Biochemical
GSK5182
Purity
>98% (HPLC)
Synonyms
GSK5182; GSK5182 biochemical
Purity/Purification
>98% (HPLC)
Target
Estrogen Receptor/ERR
Receptor
ERRgamma
NMR
Consistent with structure
Chemical Name
4-[(Z)-1-[4-(2-dimethylaminoethoxy)phenyl]-5-hydroxy-2-phenylpent-1-enyl]phenol
SMILES
CN(C)CCOc1ccc(cc1)C(c1ccc(O)cc1)=C(CCCO)c1ccccc1
Molecular Formula
C27H31NO3
CAS Number
877387-37-6
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Stability: >=2 years
Shipping: Ice Pack
Structure
Structure
Related Product Information for GSK5182 biochemical
GSK5182 is a highly selective inverse estrogen-related receptor gamma agonist (IC50: 79nM).
Product Categories/Family for GSK5182 biochemical
References
1.Kim JH et al. Estrogen-related receptor gamma is upregulated in liver cancer and its inhibition suppresses livercancer cell proliferation via induction of p21 and p27. Exp Mol Med. 2016 Mar 4; 48:e213.
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Product Notes
The GSK5182 (Catalog #AAA3611639) is a Biochemical and is intended for research purposes only. The product is available for immediate purchase. It is sometimes possible for the material contained within the vial of "GSK5182, Biochemical" to become dispersed throughout the inside of the vial, particularly around the seal of said vial, during shipment and storage. We always suggest centrifuging these vials to consolidate all of the liquid away from the lid and to the bottom of the vial prior to opening. Please be advised that certain products may require dry ice for shipping and that, if this is the case, an additional dry ice fee may also be required.Precautions
All products in the AAA Biotech catalog are strictly for research-use only, and are absolutely not suitable for use in any sort of medical, therapeutic, prophylactic, in-vivo, or diagnostic capacity. By purchasing a product from AAA Biotech, you are explicitly certifying that said products will be properly tested and used in line with industry standard. AAA Biotech and its authorized distribution partners reserve the right to refuse to fulfill any order if we have any indication that a purchaser may be intending to use a product outside of our accepted criteria.Disclaimer
Though we do strive to guarantee the information represented in this datasheet, AAA Biotech cannot be held responsible for any oversights or imprecisions. AAA Biotech reserves the right to adjust any aspect of this datasheet at any time and without notice. It is the responsibility of the customer to inform AAA Biotech of any product performance issues observed or experienced within 30 days of receipt of said product. To see additional details on this or any of our other policies, please see our Terms & Conditions page.Item has been added to Shopping Cart
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