Structure
A-836339 Biochemical
A-836339
Purity
>98% (HPLC)
Synonyms
A-836339; A836339; A-836339 biochemical
Purity/Purification
>98% (HPLC)
Suitability
DMSO: 12mg/mL
Target
Cannabinoid Receptor
Receptor
Cannabinoid Receptor
Chemical Name
Cyclopropanecarboxamide, N-[3-(2-methoxyethyl)-4, 5-dimethyl-2(3H)-thiazolylidene]-2, 2, 3, 3-tetramethyl-, [N(Z)]
SMILES
CC1=C(C)N(CCOC)/C(S1)=N/C(C2C(C)(C)C2(C)C)=O
Molecular Formula
C16H26N2O2S
CAS Number
959746-77-1
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Stability: >=2 years
Shipping: Ice Pack
Structure
Structure
Related Product Information for A-836339 biochemical
A-836339 (A836339) is a potent and selective cannabinoid CB2 receptor agonist with Ki of 0.64 and 0.76nM for human and rat CB2 receptors, displays 425- and 189-fold selectivity over CB1 receptor, respectively; exhibits full agonist efficacy (Emax=102%) with high potency (EC50=1.6nM), greater potency than other CB2-selective ligands including JWH-015 and GW-842166X; exhibits a potent CB2 receptor-mediated antihyperalgesic effect in various animal pain models, also demonstrates efficacies in the chronic constrain injury (CCI) model of neuropathic pain.
Product Categories/Family for A-836339 biochemical
References
1. Yao BB, et al. J Pharmacol Exp Ther. 2009 Jan; 328 (1):141-51.
2. McGaraughty S, et al. Neuroscience. 2009 Feb 18; 158 (4):1652-61.
3. Hsieh GC, et al. Br J Pharmacol. 2011 Jan; 162 (2):428-40.
2. McGaraughty S, et al. Neuroscience. 2009 Feb 18; 158 (4):1652-61.
3. Hsieh GC, et al. Br J Pharmacol. 2011 Jan; 162 (2):428-40.
Similar Products
Product Notes
The A-836339 (Catalog #AAA3606843) is a Biochemical and is intended for research purposes only. The product is available for immediate purchase. It is sometimes possible for the material contained within the vial of "A-836339, Biochemical" to become dispersed throughout the inside of the vial, particularly around the seal of said vial, during shipment and storage. We always suggest centrifuging these vials to consolidate all of the liquid away from the lid and to the bottom of the vial prior to opening. Please be advised that certain products may require dry ice for shipping and that, if this is the case, an additional dry ice fee may also be required.Precautions
All products in the AAA Biotech catalog are strictly for research-use only, and are absolutely not suitable for use in any sort of medical, therapeutic, prophylactic, in-vivo, or diagnostic capacity. By purchasing a product from AAA Biotech, you are explicitly certifying that said products will be properly tested and used in line with industry standard. AAA Biotech and its authorized distribution partners reserve the right to refuse to fulfill any order if we have any indication that a purchaser may be intending to use a product outside of our accepted criteria.Disclaimer
Though we do strive to guarantee the information represented in this datasheet, AAA Biotech cannot be held responsible for any oversights or imprecisions. AAA Biotech reserves the right to adjust any aspect of this datasheet at any time and without notice. It is the responsibility of the customer to inform AAA Biotech of any product performance issues observed or experienced within 30 days of receipt of said product. To see additional details on this or any of our other policies, please see our Terms & Conditions page.Item has been added to Shopping Cart
If you are ready to order, navigate to Shopping Cart and get ready to checkout.
