Structure
L 888607, Inhibitor | L888607, inhibitor
L 888607
Purity
98.00%
Synonyms
L 888607; L888607; inhibitor
Purity/Purification
98.00%
Form/Format
Solid. Powder
Solubility
DMSO: 150mg/mL (399.11mM)
(<1mg/ml refers to the product slightly soluble or insoluble)
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C19H15ClFNO2S
SMILES
O=C(O)C[C@@H]1CCN2C1=C(SC3=CC=C(Cl)C=C3)C4=C2C=C(F)C=C4
CAS Number
860033-06-3
Target & IC50
CRTH2/DP2 Receptor: ic50 0.8nM (ki)
TP Receptor: ic50 283nM (ki)
DP/DP1 Receptor: ic50 2331nM (ki)
EP2 Receptor: ic50 8748nM (ki)
EP3-III Receptor: ic50 1260nM (ki)
EP4 Receptor: ic50 4634nM (ki)
FP Receptor: ic50 10018nM (ki)
IP Receptor: ic50 14434nM (ki)
TP Receptor: ic50 283nM (ki)
DP/DP1 Receptor: ic50 2331nM (ki)
EP2 Receptor: ic50 8748nM (ki)
EP3-III Receptor: ic50 1260nM (ki)
EP4 Receptor: ic50 4634nM (ki)
FP Receptor: ic50 10018nM (ki)
IP Receptor: ic50 14434nM (ki)
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
-80 degree C for 2 years in solvent
Structure
Structure
Related Product Information for L888607, inhibitor
L 888607 is an effective and selective CRTH2 agonist (Ki: 0.8nM).
Product Categories/Family for L888607, inhibitor
References
Gervais FG, Identification of a potent and selective synthetic agonist at the CRTH2 receptor. Mol Pharmacol. 2005 Jun;67(6):1834-9.
Similar Products
Product Notes
The L888607 (Catalog #AAA5755150) is an Inhibitor and is intended for research purposes only. The product is available for immediate purchase. It is sometimes possible for the material contained within the vial of "L 888607, Inhibitor" to become dispersed throughout the inside of the vial, particularly around the seal of said vial, during shipment and storage. We always suggest centrifuging these vials to consolidate all of the liquid away from the lid and to the bottom of the vial prior to opening. Please be advised that certain products may require dry ice for shipping and that, if this is the case, an additional dry ice fee may also be required.Precautions
All products in the AAA Biotech catalog are strictly for research-use only, and are absolutely not suitable for use in any sort of medical, therapeutic, prophylactic, in-vivo, or diagnostic capacity. By purchasing a product from AAA Biotech, you are explicitly certifying that said products will be properly tested and used in line with industry standard. AAA Biotech and its authorized distribution partners reserve the right to refuse to fulfill any order if we have any indication that a purchaser may be intending to use a product outside of our accepted criteria.Disclaimer
Though we do strive to guarantee the information represented in this datasheet, AAA Biotech cannot be held responsible for any oversights or imprecisions. AAA Biotech reserves the right to adjust any aspect of this datasheet at any time and without notice. It is the responsibility of the customer to inform AAA Biotech of any product performance issues observed or experienced within 30 days of receipt of said product. To see additional details on this or any of our other policies, please see our Terms & Conditions page.Item has been added to Shopping Cart
If you are ready to order, navigate to Shopping Cart and get ready to checkout.
