Z-VAD-FMK, Inhibitor

Z-VAD-FMK

Cat. Num. AAA385773

• Purity: >98%
• Synonyms: Z-VAD-FMK; inhibitor

• Purity/Purification: >98%
• Form/Format: Powder
• Concentration: 0.1 mM: 21.39 mL (1 mg); 106.95 mL (5 mg); 213.91mL (10 mg); 0.5 mM: 4.28 mL (1 mg); 21.39 mL (5 mg); 42.78 mL (10 mg); 1 mM: 2.14 mL (1 mg); 10.7 mL (5 mg); 21.39 mL (10 mg); 5 mM: 0.43 mL (1 mg); 2.14 mL (5 mg); 4.28 mL (10 mg) (varies by lot)

• CAS Number: 187389-52-2
• Formula: C22H30FN3O7
• SMILES: C[C@@H](C(=O)N[C@@H](CC(=O)OC)C(=O)CF)NC(=O)[C@H](C(C)C)NC(=O)OCC1=CC=CC=C1
• Actions: Inhibitor
• In Vivo Solvent: DMF
• Solubility (DMSO): 93 mg/mL (198 mM)
• Solubility (Ethanol): 24 mg/mL heating (51 mM)
• Solubility (in vivo): 84 mg/mL
• Solubility (Water): <1 mg/mL (<1 mM)
• Availability: We cannot ship this item to Switzerland, Italy, Germany, France and Austria.
• Preparation and Storage: at -20 degree C 3 years Powder

Chemical Structure

Related Product Information for Z-VAD-FMK, inhibitor

Z-VAD-FMK is a cell-permeable, irreversible pan-caspase inhibitor. Inhibits caspase processing and apoptosis induction in tumor cells in vitro (IC50 = 0.0015 - 5.8 mM). Active in vivo.

References

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